| Description | ACTIVE HALF-LIFE 5-7 Days
TABLET COUNT: 50 COUNTS
CLASSIFICATION SERM
DOSAGE 50-100 mg/day
ACNE No
WATER RETENTION No
HBR Rare
HEPATOTOXICITY Low
AROMATIZATION No | Tablet Count: 100 tablets
Dose: 20– 60mcg per day
Cycle: 6-8 weeks.
Bioavailability: 89–98% (orally)
Molar mass: 277.19
Elimination half-life: 36–48 hours
Metabolism: Hepatic (negligible)
Acne: RARELY
Water Retention: RARELY
HBR: NO
Hepatoxity: LOW
Aromatization: YES | ACTIVE INGREDIENT: Exemestane 25 mg
TABLET COUNT: 30 COUNTS
ACTIVE HALF-LIFE: 9 HOURS
CLASSIFICATION: ANABOLIC STEROID
DOSAGE MEN: 25-50 MG/DAY
DOSAGE WOMEN: 5-30 MG/DAY
ACNE: RARELY
WATER RETENTION: NO
HBR: NO
HEPATOXITY: LOW
Ship From: Europe | Product Name: Halotestin 10mg
Active Ingredient: Fluoxymesterone 10mg
Active Life: 9 Hours
Drug Class: Androgen; Anabolic Steroid
Detection Time: 11 Months
Common Doses: 10-20 mg/day
Blood pressure: Perhaps
Acne: Yes
Water retention: No
Aromatisation: No
Liver toxicity: High
Decrease HPTA function: None | ACTIVE INGREDIENT: LETROZOLE 5mg
TABLET COUNT: 100 COUNTS
ACTIVE HALF-LIFE: 9 HOURS
CLASSIFICATION: ANTI ESTROGEN
DOSAGE: 5mg
ACNE: NONE
WATER RETENTION: NO
HBR: NO
HEPATOXITY: LOW
AROMATIZATION: NO | Active Ingredient: Exemestane 25 Mg
Tablet Count: 25 Counts
Active Half-life: 9 Hours
Classification: Anabolic Steroid
Dosage Men: 25-50 Mg/day
Dosage Women: 5-30 Mg/day
Acne: Rarely
Water Retention: No
Hbr: No
Hepatoxity: Low |
| Content | Clomixin – a synthetic estrogen, which is usually assigned to women that have difficulty conceiving a child. As for men, the application of Clomiphene Citrate increases the level of hormones that stimulate the testicles. That is Clomixin acts directly on the pituitary gland. This increases the natural production of testosterone by the body.
Chemically for athletes this is highly a favorable effect, since at the end of cycle Testosterone levels are higher than normal. Once the athlete stops taking medication, testosterone levels significantly decreased and its natural level must be returned. Because of this, there are considerable loss of muscle mass and volume. Studies show that when taking Clomiphene Citrate in the amount of 50-100 mg per day, in the evening or in the morning, after meals, in the two-week period or more natural testosterone production is back to normal.
Clomixin Effects
During the period of Clomixin use, it raises testosterone levels. As effective is Clomixin as an anti-estrogen. Many athletes experience a surplus in it after completing the cycle. A high level of the hormone in combination with low testosterone may lead to the development of gynecomastia. Clomixin – solves two problems: blocks unwanted effect of estrogen; rising natural level of testosterone in the body.
In this regard as of side effects, it is considered a fairly safe drug. Clomixin is both women and men, in that there are no contraindications. Women who use this drug helps to achieve tighter appearance before the competition. There may be temporary visual disturbances.
How to Use Clomixin: Dosage, Cycle, Reviews
In the early cycle apply two tablets a day (it is 100 mg). Then, the dosage can go to one tablet per day.
Warnings: Keep out of reach of children. For adults only. | Clenbuterol hydrochloride 0.02mg x 100 tablets
Clenbuterol is a widely used bronchodilator in many parts of the world. The drug is most often prepared in 20mcg tablets, but it is also available in syrup and injectable form. Clenbuterol belongs to a broad group of drugs knows as sympathomimetics. | Exemestane is a synthetic androgen analogue. It’s is a steroidal inhibitor of aromatase which binds irreversibly to and inhibits the enzyme aromatase, thereby blocking the conversion of cholesterol to pregnenolone and the peripheral aromatization of androgenic precursors into estrogens.
Exemestane has been associated with a low rate of serum enzyme elevations during therapy and rare instances of clinically apparent liver injury.
This medication is used to treat certain types of breast cancer (such as hormone-receptor-positive breast cancer) in women after menopause. Exemestane is also used to help prevent the cancer from returning. Some breast cancers are made to grow faster by a natural hormone called estrogen. Exemestane decreases the amount of estrogen the body makes and helps to slow or reverse the growth of these breast cancers. Exemestane is usually not used in women of childbearing age.
Exemestane is usually taken once a day after a meal. Take Exemestane at around the same time every day. You may need to take Exemestane for several years or longer. Continue to take Exemestane even if you feel well. Do not stop taking Exemestane without talking to your doctor.
Effect On Estrogens
Plasma estrogen (estradiol, estrone, and estrone sulfate) suppression is seen starting at a 5-mg daily dose of Exemestane, with a maximum suppression of at least 85% to 95% achieved at a 25-mg dose. Exemestane 25 mg daily reduces whole body aromatization (as measured by injecting radiolabeled androstenedione) by 98% in postmenopausal women with breast cancer. After a single dose of Exemestane 25 mg, the maximal suppression of circulating estrogens occurres 2 to 3 days after dosing and persisted for 4 to 5 days.
Effect On Corticosteroids
In multiple-dose trials of doses up to 200 mg daily, Exemestane selectivity was assessed by examining its effect on adrenal steroids. Exemestane did not affect cortisol or aldosterone secretion at baseline or in response to ACTH at any dose. Thus, no glucocorticoid or mineralocorticoid replacement therapy is necessary with Exemestane treatment.
Other Endocrine Effects
Exemestane does not bind significantly to steroidal receptors, except for a slight affinity for the androgen receptor (0.28% relative to dihydrotestosterone). The binding affinity of its 17dihydrometabolite for the androgen receptor, however, is 100 times that of the parent compound.
Daily doses of Exemestane up to 25 mg had no significant effect on circulating levels of androstenedione, dehydroepiandrosterone sulfate, or 17-hydroxyprogesterone, and were associated with small decreases in circulating levels of testosterone.
Increases in testosterone and androstenedione levels have been observed at daily doses of 200 mg or more. A dose-dependent decrease in sex hormone binding globulin (SHBG) has been observed with daily Exemestane doses of 2.5 mg or higher.
Slight, nondose-dependent increases in serum luteinizing hormone (LH) and follicle-stimulating hormone (FSH) levels have been observed even at low doses as a consequence of feedback at the pituitary level. Exemestane 25 mg daily had no significant effect on thyroid function [free triiodothyronine (FT3), free thyroxine (FT4), and thyroid stimulating hormone (TSH).
Absorption
Exemestane is distributed extensively into tissues. Exemestane is 90% bound to plasma proteins and the fraction bound is independent of the total concentration. Albumin and α11-acid glycoprotein both contribute to the binding. The distribution of Exemestane and its metabolites into blood cells is negligible.
Metabolism
Exemestane is extensively metabolized. The initial steps in the metabolism of Exemestane are oxidation of the methylene group in position 6 and reduction of the 17-keto group with subsequent formation of many secondary metabolites.
Each metabolite accounts only for a limited amount of drug-related material. The metabolites are inactive or inhibit aromatase with decreased potency compared with the parent drug. One metabolite may have androgenic activity [see Pharmacodynamics]. Studies using human liver preparations indicate that cytochrome P 450 3A4 (CYP 3A4) is the principal isoenzyme involved in the oxidation of Exemestane. Exemestane is metabolized also by aldoketoreductases. | Fluoxymesterone 10mg x 100 tablets
Fluoxymesterone has established itself as a high-quality drug with a high androgenic index. Fluoxy mesteronegives a great increase in strength. Suitable for preparation for competitions, when an athlete needs strength without a large set of muscle mass. In this case, the musculature gets the necessary hardness. | Letrozole 5mg x 100 tablets
Letrozole is a third generation Aromatase Inhibitor (AI) that works by attaching to -and eliminating the aromatase enzyme resposible for producing estrogen. This makes it a perfect choice to combat gynocomastia which it will completely prevent. Letrozole also quite raises LH levels which deems it suitable for post-cycle use. The human body does need estrogen to maintain proper immune function and balance cholesterol ratios in the blood. Since letrozole is so strong at eliminating estrogen, it is not suited for long term use. | |
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